potent macrocyclic PCSK9 PPI inhibitor
1000x optimization of biochem. activity
from mRNA display screen and SBDD
J. Med. Chem., 2020, Nov. 10, 2020
Merck, PA + NJ / UCB Ra Pharma, MA
Merck/UCB/Ra Pharma macrocyclic PCSK9 protein-protein interaction (PPI) inhibitor