oral TRPV4 ion channel antagonist backup
proj. human dose <100 mg QD for pul. edema
backup to GSK2798745 / GSK3527497
J. Med. Chem., Nov. 17, 2020
GlaxoSmithKline, Collegeville, PA
“compound 36” (GlaxoSmithKline (GSK) oral TRPV4 ion channel antagonist backup)