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Sep. 18, 2021

DS-1971a: A potent, Isoform-Selective Arylsulfonamide NaV1.7 Inhibitor

DS-1971a

potent, selective NaV1.7 ion channel inhibitor completed Ph. I in HV, discontinued in Ph. II from optimization of known starting point J. Med. Chem., May 26, 2020 Daiichi Sankyo, Tokyo, JP

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