Genentech ER Degrader
selective ER degrader (SERD) + full antag. oral (30 mg QD), Ph. III for ER+, HER2- BC from profiling >4k cmpds for desired MoA giredestrant (GDC-9545) Genentech, South San Francisco, CA
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- Genentech ER Degrader
- Pfizer CoV-2 MPro Inhibitor
- Arvinas ER Chimeric Degrader
- Kronos CDK9 Inhibitor
- Merck PCSK9 Inhibitors
- Mirati KRASG12D Inhibitor
- Takeda EGFRex20 Inhibitor
- Lilly GLP Molecular Glue
- RevMed KRASG12C Tricomplex Inhibitor
- Genentech mPI3Kα Degrader
- H3Bio SF3b Splicing Modulator
- BioCryst Kallikrein Inhibitor
- Genentech ER Degrader