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Sep. 13, 2024

An Orally Bioavailable TGFβ Type I Receptor Kinase Inhibitor

vactosertib

TGFβ type I receptor inhibitor Ph. II in oncology from literature compound, opt. of kinase selectivity and PK properties Nat. Commun., August 2024 Ewha Womans University, Seoul, KR; Medpacto, Seoul, KR

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