A Dual 5-HT2A and 5-HT2C Receptor Inverse Agonist Developed to Address the Limitations of Pimavanserin
compound 8
5-HT2A/5-HT2C receptor inverse agonist preclinical in dementia-related psychosis pimavanserin lead, SBDD, hERG liability, and microsomal stability opt. J. Med. Chem., August 2024 Shionogi Pharmaceutical Research Center, Osaka, JP; Kyoto University, Kyoto, JP
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