Unexpected KRAS(G12C)(ON) Inhibition by BridgeBio's Covalent Clinical Compound
BBO-8520
oral covalent KRAS(G12C)(ON/OFF) inhibitor Ph. I for advanced non-small cell lung cancer from known inhibitor AACR Annual Meeting 2024, San Diego, CA BridgeBio, San Francisco, CA / NCI RAS Initiative, Frederick, MD
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vactosertib
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casdatifan (AB521)
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bomedemstat (MK-3543, IMG-7289)
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