< 1 minute read
Sep. 17, 2021

Tucatinib: EGFR-Sparing HER2 Kinase Inhibitor

tucatinib

EGFR-sparing HER2 kinase inhibitor approved in met. HER2+ BC incl. w/ brain met. from optimization of known TKIs Mol. Cancer Ther., Apr. 1, 2020 Array / Cascadian Tx / Seattle Genetics

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