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Sep. 18, 2021
TNO155: A First-in-Class Allosteric SHP2 Phosphatase Inhibitor
TNO155
first-in-class allosteric SHP2 phosphatase inh. oral agent in multiple trials for cancer from 1.5M cmpd biochemical HTS + SBDD J. Med. Chem., Sep. 24, 2020 Novartis, Cambridge, MA