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Sep. 18, 2021

EST73502: A Dual µ-Opioid Receptor Agonist, σ1 Antagonist

"EST73502"

dual µ-opioid receptor agonist, σ1 antagonist oral analgesia w/ reduced opioid AEs, in Ph. I from literature cmpd pharmacophore merging J. Med. Chem., Oct. 16, 2020 ESTEVE Pharmaceuticals SA, Barcelona, ES

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