< 1 minute read
Dec. 10, 2021

SJ995973: A Bifunctional Degrader

compound 4c

degrader with simpler CRBN warhead BRD4 DC50 = 0.87 nM, Dmax = 99% from structure-based design Angewandte Chemie Int. Ed. Saint Jude Children’s Hospital, Memphis, TN

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