SJ995973: A Bifunctional Degrader
compound 4c
degrader with simpler CRBN warhead BRD4 DC50 = 0.87 nM, Dmax = 99% from structure-based design Angewandte Chemie Int. Ed. Saint Jude Children’s Hospital, Memphis, TN
degrader with simpler CRBN warhead BRD4 DC50 = 0.87 nM, Dmax = 99% from structure-based design Angewandte Chemie Int. Ed. Saint Jude Children’s Hospital, Memphis, TN