Compound 10: A TGFβR Inhibitor Prodrug
compound 10
tumor specific prodrug of TGFβR inhibitor QW dosing, improved tumor-to-heart ratio BMS-986260 prodrug w/ self-immolative link. Journal of Medicinal Chemistry Bristol Myers Squibb, Princeton, NJ
tumor specific prodrug of TGFβR inhibitor QW dosing, improved tumor-to-heart ratio BMS-986260 prodrug w/ self-immolative link. Journal of Medicinal Chemistry Bristol Myers Squibb, Princeton, NJ