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Dec. 10, 2021
Aficamten: Next-Generation Myosin Inhibitor
aficamten
oral QD myosin inhibitor (IC50 = 1.4 µM) Ph. II candidate for cardiomyopathy (5-30 mg) from HTS w/ bovine cardiac muscle myofibrils Journal of Medicinal Chemistry Cytokinetics, South San Francisco, CA