2022
- resmetirom
- RMC-5552
- inavolisib
- BI 685509
- DN-1289
- paltusotine
- SPR720
- emraclidine
- compound 25
- compound 49
- sebetralstat
- GDC-2394
- compound 5g
- AZD1656
- JNJ-64264681
- BI-0474
- compound 57
- AN15368
- UCB7362
- BAY-069
- compound 3
- compound 19
- compound 23
- obicetrapib
- ACT-660602
- compound 7
- SPH3127
- AZD4831
- compound 6
- GNE-064
- Compound 33
- RP-6306
- BLU-945
- SAGE-718
- BI-4142
- CHF-6366
- Compound 3f
- MRTX0902
- Compound 14
- CC-99677
- Compound 23
- BMS-986120
- EZM0414
- DNL201
- Iclepertin
- BMS-986339
- MK-0159
- TAS1553
- NTQ1062
- Apararenone
- Pevonedistat
- Compound 20
- NVP-CLR457
- TXA6101
- RLX-33
- INCB13739
- Compound 4e
- MAGLi 43
- Sudapyridine (WX-081)
- Dorzagliatin
- JDQ443
- AZD4625
- JBJ-09-063
- ABBV-318
- tenapanor
- lenrispodun
- compound 41
- DS69910557
- compound 14
- compound 53