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A Covalent Allosteric WRN Helicase Inhibitor Stemming from Chemoproteomics Screening

VVD-214/RO7589831

oral, covalent, allosteric WRN helicase inhibitor Ph. I for MSI and/or dMMR advanced solid tumors chemoproteomics screening technology AACR Annual Meeting 2024 New Drugs on the Horizon Vividion Therapeutics, San Diego, CA / Roche, Basel, CH

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