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Apr. 19, 2022
Rilzabrutinib: A Billion-Dollar Reversible Covalent Inhibitor from Principia
rilzabrutinib (PRN1008)
oral reversible covalent BTK inhibitor in Ph. III for immune thrombocytopenia from structure-based drug design + opt. J. Med. Chem., March 18, 2022 Principia Biopharma (Sanofi), So. San Francisco, CA
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