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Dec. 16, 2021

PTC596: a Brain-Penetrant Tubulin-Binding Agent

PTC596

CNS-penetrant tubulin-binder (colchicine site) oral agent in Ph. I for leiomyosarcoma not a P-gp substrate, formerly BMI-1 inh. Molecular Cancer Therapeutics PTC Therapeutics, South Plainfield, US

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