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Dec. 16, 2021

Giredestrant: Oral Selective Estrogen Receptor Degrader (SERD) and Full Antagonist

giredestrant

selective ER degrader (SERD) + full antagonist oral (30 mg QD), Ph. III for ER+, HER2- BC from profiling >4k cmpds for desired MoA Journal of Medicinal Chemistry Genentech, San Francisco, US

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