Apr. 19, 2022

MAK683: A Pioneering EZH2/PRC2 Inhibitor in Oncology

MAK683

oral, allosteric PRC2 inhibitor (EED) in Ph. I/II for cancer (DLBCL); preliminary efficacy from micromolar HTS hit J. Med. Chem., March 30, 2022 Novartis, Emeryville, CA

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