< 1 minute read
Nov. 26, 2021
GSK3685032: A First-In-Class DNMT1 Inhibitor
GSK3685032
selective rev. DNA methyltransferase inhibitor preclinical eff. at 30 mpk SC BID (xenograft) from 1.8M cmpd enzymatic HTS + opt. Nature Cancer GlaxoSmithKline
selective rev. DNA methyltransferase inhibitor preclinical eff. at 30 mpk SC BID (xenograft) from 1.8M cmpd enzymatic HTS + opt. Nature Cancer GlaxoSmithKline