< 1 minute read
Nov. 26, 2021

GSK3685032: A First-In-Class DNMT1 Inhibitor

GSK3685032

selective rev. DNA methyltransferase inhibitor preclinical eff. at 30 mpk SC BID (xenograft) from 1.8M cmpd enzymatic HTS + opt. Nature Cancer GlaxoSmithKline

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