>50x family-selective CDK9 kinase inhibitor

IV agent (5-30 mg QW) in Ph. I for cancer

scaffold hop from atuveciclib

Journal of Medicinal Chemistry

Bayer, Berlin, DE / Vincerx, Palo Alto, US

The Vincerx Pharma/Bayer CDK9 inhibitor, VIP152 (BAY 1251152), is a once-weekly (5-30 mg) IV agent in Ph. I for cancer with >50x family-selectivity. The sulfoximine-containing molecule is derived from the oral…


 become a member to continue reading

Ask your company or librarian about a Drug Hunter membership to to see all summaries and get access to even more helpful information.

  • Stay up-to-date and save more time with exclusive members-only content
  • On-board new team members with educational content and case studies
  • Generate ideas and discussion with easy-to-read slide decks
  • Generate ideas and discussion with easy-to-read slide decks