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Jan. 28, 2023

Inavolisib: An Isoform-Selective Mutant PI3Ka Monovalent Degrader

inavolisib

isoform-selective mutant PI3Kα degrader oral <9 mg QD, Ph. III in HR+/HER2- BC from cellular characterization of PI3Ki and opt. J. Med. Chem., December 1, 2022 Genentech, South San Francisco, CA

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