allosteric mutant-selective IDH1 inhibitor
oral, in clinical development
from SBDD of prior mIDH inhibitor
J. Med. Chem. 2020, 63, 1612-1623
FORMA Therapeutics, Watertown, MA
FT-2102 (olutsidenib) (FORMA oral allosteric mutant-selective IDH1 inhibitor clinical candidate)