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Sep. 18, 2021

CVN424: A CNS Penetrant GPR6 GPCR Inverse Agonist

CVN424

CNS pen. GPR6 GPCR inverse agonist oral QD Ph. II candidate for Parkinson's from 360k cmpd cell-based HTS + opt. J. Pharmacol. Exp. Ther., Apr. 1, 2021 Cerevance / Takeda California, San Diego, US

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