< 1 minute read
Jan. 17, 2022

RP-3500 is an Oral ATR Kinase Inhibitor

RP-3500

ATR kinase inhibitor phase I/IIa candidate for advanced solid tumors from lipid-kinase inhibitor scaffold Molecular Cancer Therapeutics Repare Therapeutics, Saint-Laurent, CAN

drughunter.com
Drug Hunter Team

RP-3500 is an oral ATR kinase inhibitor and Ph. II clinical candidate for advanced solid tumors with ATRi-sensitizing mutations, alone or in combination with talazoparib (PARPi) or gemcitabine. Reviewer Anthony Vaganos says, “An ATR molecule ( ceralasertib ) is in clinical trials but studies in two different tumors in combination with PARP [...]

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