Jun. 4, 2023
Roginolisib: The First Clinical Non-Competitive PI3Kd Inhibitor
IOA-244 (roginolisib)
oral QD non-competitive PI3Kd inhibitor Ph. I in metastatic cancers from focused kinase inhibitor screen (60K cmpds) + opt. Cancer Res. Commun., April 14, 2023 Merck Serono / iOnctura, CH