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May 9, 2023

Roblitinib is an Orally Available Aldehyde Selective for FGFR4

FGF401 (roblitinib)

oral reversible-covalent FGFR4 kinase inhibitor first sel. FGFR4i in clinical studies; for HCC from biochemical HTS and SBDD J. Med. Chem., Oct. 1, 2020 Novartis, Basel, CH

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