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lead finding

  • Cover image of Drug Hunter article "Where Do Recent Small Molecule Clinical Candidates Come From?"

    Where Do Recent Small Molecule Clinical Candidates Come From?

    Modern hit-finding technologies are incredible. Dean Brown and Jonas Bostrom at AstraZeneca have a very nice review out summarizing the hit-finding strategies for 66 clinical candidates published from 2016-2017. Some highlights include a clinical candidate from DNA-encoded libraries at GSK, the discovery of an RNA-binding drug candidate by PTC/Roche, and fragment-based programs with candidates 100,000x…

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  • Molecules
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© Rosalind Scientific LLC 2018-2022