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  • Solid Form Strategies for Increasing Oral Bioavailability

    Small-molecule drug candidates are increasingly falling “beyond the rule of 5,” making oral administration more challenging. Optimizing a drug’s solid form can improve its solubility and bioavailability when further molecular modifications are prohibitive. This minireview covers solid form strategies for increasing the solubility and oral bioavailability of small-molecule drugs including: Cryo-milling Salt formation Spray drying…

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  • Molecules
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  • Find Partners
    • Drug Discovery CROs
    • Drug Development CDMOs
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    • Drug Discovery Companies
    • Drug Discovery Investors
  • Premium
  • Advisory Board
  • Our Reviewers
  • About Us
  • Sponsors
  • Advertise
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  • Our Team
  • Blog
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  • LinkedIn
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© Rosalind Scientific LLC 2018-2022