Drug Hunter’s February 2022 Small Molecules of the Month include a glucokinase partial activator, an orexin receptor agonist intended to promote wakefulness rather than sleep, and an orally available diacid, among others.
Is BMS-820132 a prodrug?
How is T-690 different from previous generations of GCS inhibitors?
Which off-target is correlated to loss of appetite in rats?
What were the starting points for these molecules?
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