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molecules of the month

December 2021

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Drug Hunter Molecules of the Month December 2021 1. MRTX1133 – Mirati KRAS G12D Inhibitor 2. CC-90001 – BMS c-Jun N-Terminal Kinase Inhibitor CC-90001 3. HTT-D3 – PTC Therapeutics HTT-lowering splicing modifier 4. ulotaront – TAAR1 agonist 5. velsecorat – AstraZeneca inhaled glucocorticoid receptor modulator 6. “compound 22” – Vertex ether-based ELOVL1 inhibitors 7. “compound 43b” – Takeda RBP4 reducer 8. RP-3500 – Repare Therapeutics ATR inhibitor 9. HR011303 – Jiangsu Hengrui URAT1 inhibitor 10. “compound 54c” – GSK inhaled JAK1 inhibitor 11. “compound 17a” – Sanofi SGK1 inhibitor 12. “compound 3” – Pfizer Vanin-1 inhibitor 13. “compound 24” – Merck LRRK2 inhibitor 14. “compound 25” – Genentech HPK1 inhibitor

The December edition of Small Molecules of the Month includes a Ph. III candidate identified from machine-learning-assisted in vivo phenotypic screening, Mirati’s KRAS G12D inhibitor, and several kinase inhibitors outside of oncology.

Thanks to reviewers Joachim Rudolph, Naomi Rajapaksa, Julien Lefranc, Christian Kuttruff, Christian Gampe, Jake Schwarz, Yoana Dimitrova, Anthony Vaganos, and Kim Huard for their nominations and key insights this month.

Premium subscribers can read details behind each molecule and download the slide deck. Sign up for the free e-mail newsletter to get a preview each month.

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Slide Deck - Small Molecules of the Month - December 2021
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