“PROTAC 6”

IAP-based selective RIPK2 degrader

prolonged PD w/ 0.15 mpk SC Q3D dosing

E3 binder switch and property-based opt.

Commun. Biol., Mar. 20, 2020

GlaxoSmithKline, Stevenage, UK / PMCC

“PROTAC 6” (GlaxoSmithKline (GSK) IAP-based selective RIPK2 degrader with prolonged in vivo PD)


 become a member to continue reading

Ask your company or librarian about a Drug Hunter membership to to see all summaries and get access to even more helpful information.

  • Stay up-to-date and save more time with exclusive members-only content
  • On-board new team members with educational content and case studies
  • Generate ideas and discussion with easy-to-read slide decks
  • Generate ideas and discussion with easy-to-read slide decks