Gout is caused by the buildup of uric acid. The main treatments are drugs that increase uric acid secretion (uricosurics, e.g. probenecid ) and xanthine oxidase inhibitors which inhibit uric acid production (e.g. allopurinol ). URAT1 inhibitors like lesinurad (Ironwood Pharmaceuticals) and dotinurad are emerging treatments, inhibiting uric [...]
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Jan. 17, 2022
HR011303 is a URAT1 Inhibitor for Gout
HR011303
human uric acid transporter inhibitor phase III candidate for hyperuricemia and gout from pharmacophore-based lead generation Drug Metabolism and Disposition Jiangsu Hengrui Medicine Co., Shanghai, CN