dual _-opioid receptor agonist, _1 antagonist
oral analgesia w/ reduced opioid AEs, in Ph. I
from literature cmpd pharmacophore merging
J. Med. Chem., Oct. 16, 2020
ESTEVE Pharmaceuticals SA, Barcelona, ES
“EST73502”
1 min read
“EST73502” (ESTEVE oral dual mu-opioid receptor agonist, sigma-1 receptor antagonist clinical candidate)
Search By Structure
- BAY 1214784
- BAY 1217224
- CC-90011
- LEO 39652
- OATD-01
- AG-636
- “compound 46”
- “compound 25”
- “lipid 10a”
- BAY-6672
- “compound 27”
- “EST73502”
- CG428
- “compound 34”
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