Nov. 28, 2022

Roche's Allosteric EGFR(L858R) Inhibitor and Degrader Progenitor

compound 57

oral EGFRL858R inhibitor efficacy in EGFR mutant mouse models SBDD opt. from previously disclosed EGFRai J. Med. Chem. F. Hoffmann-La Roche, Basel, CH

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