AG-881 (vorasidenib) (Agios oral brain penetrant allosteric mutant IDH1/2 dual inhibitor clinical candidate)
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Sep. 15, 2021
AG-881: An oral brain penetrant allosteric mutant IDH1/2 dual inhibitor clinical candidate
AG-881
allosteric mutant IDH1/2 dual inhibitor oral, brain penetrant, completed Ph. I in HV from SBDD of prior mIDH inhibitor ACS Med. Chem. Lett., 2020, 11, 101-107 Agios Pharmaceuticals, Cambridge, MA