Sep. 18, 2021

ACT-1004-1239: A CXCR7 GPCR Insurmountable Antagonist

ACT-1004-1239

CXCR7 GPCR insurmountable antagonist target engagement in rodent, 61% F in dog from 300k HTS vs. β-arrestin recruitment, opt. J. Med. Chem., Dec. 14, 2020 Idorsia Pharma (Actelion), Allschwil, CH

drughunter.com
Drug Hunter Team

Idorsia/Actelion CXCR7 GPCR insurmountable antagonist

Loading...

twitterlinkedinemail

Other molecules you may be interested in